5-HT4 receptor

• BIMU-8
• Cisaprid
• CJ-033,466
• Mosaprid
• Prukaloprid
• Renzaprid
• RS-67506
• RS-67333 - parcijalni agonist
• SL65.0155 - parcijalni agonist
• Tegaserod
• Zakoprid

Antagonisti

• Piboserod
• GR-113,808 (1-metil-1H-indol-3-karboksilna kiselina, [1-[2-[(metilsulfonil)amino]etil]-4-piperidinil]metil ester)^[10]
• GR-125,487
• RS-39604 (1-[4-Amino-5-hloro-2-(3,5-dimetoksifenil)metiloksi]-3-[1-[2-metilsulfonilamino]piperidin-4-il]propan-1-on)
• SB-203,186
• ([Metoksi-¹¹C]1-butilpiperidin-4-jil)metil 4-amino-3-metoksibenzoat^[11]

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2. ^ Blondel O, Vandecasteele G, Gastineau M, Leclerc S, Dahmoune Y, Langlois M, Fischmeister R (1997). „Molecular and functional characterization of a 5-HT4 receptor cloned from human atrium.” (PDF). FEBS Lett. 412 (3): 465—74. PMID 9276448. S2CID 23714426. doi:10.1016/S0014-5793(97)00820-X. CS1 одржавање: Вишеструка имена: списак аутора (веза)^{[мртва веза]}
3. ^ „Entrez Gene: HTR4 5-hydroxytryptamine (serotonin) receptor 4”. Приступљено 1. 7. 2018. 
4. ^ Hegde, SS; Eglen, RM (1. 10. 1996). „Peripheral 5-HT4 receptors”. The FASEB Journal. 10 (12): 1398—1407. PMID 8903510. S2CID 21596751. doi:10.1096/fasebj.10.12.8903510.  Пронађени су сувишни параметри: |author= и |last1= (помоћ); Пронађени су сувишни параметри: |author2= и |last2= (помоћ)
5. ^ Katarina Varnäs, Christer Halldin, Victor W. Pike; Håkan Hall (2003). „Distribution of 5-HT₄ receptors in the postmortem human brain–an autoradiographic study using [¹²⁵]SB 207710”. European Neuropsychopharmacology. 13 (4): 228—234. PMID 12888181. S2CID 27945284. doi:10.1016/S0924-977X(03)00009-9. CS1 одржавање: Вишеструка имена: списак аутора (веза)
6. ^ Mnie-Filali, O.; Amraei, M. G.; Benmbarek, S.; Archer-Lahlou, E.; Peñas-Cazorla, R.; Vilaró, M. T.; Boye, S. M.; Piñeyro, G. (2010). „Serotonin 4 receptor (5-HT4R) internalization is isoform-specific: Effects of 5-HT and RS67333 on isoforms a and B”. Cellular Signalling. 22 (3): 501—509. PMID 19922792. doi:10.1016/j.cellsig.2009.11.004. 
7. ^ Pellissier LP, Sallander J, Campillo M, Gaven F, Queffeulou E, Pillot M, Dumuis A, Claeysen S, Bockaert J, Pardo L (2009). „Conformational toggle switches implicated in basal constitutive and agonist-induced activated states of 5-hydroxytryptamine-4 receptors” (PDF). Molecular Pharmacology. 75 (4): 982—90. PMID 19168624. S2CID 17957338. doi:10.1124/mol.108.053686. 
8. ^ Kornum, B. R.; N. M. Lind; N. Gillings; Marner, Lisbeth; F. Andersen; Gitte Moos Knudsen (2008). „Evaluation of the novel 5-HT(4) receptor PET ligand [(11)C]SB207145 in the Gottingen minipig”. Journal of Cerebral Blood Flow and Metabolism. 29 (1): 186—196. PMID 18797470. S2CID 16196384. doi:10.1038/jcbfm.2008.110. 
9. ^ Lisbeth Marner, Nic Gillings, Roger Gunn, Robert Comley, William Baaré, Steen Hasselbalch and Gitte Knudsen (1. 5. 2008). „Quantification of 11C-SB207145-PET for 5-HT4 receptors in the human brain: Preliminary results”. Journal of Nuclear Medicine. 48 (Supplement 2) (Supplement 2): 159P. Архивирано из оригинала 3. 3. 2016. г. Приступљено 24. 7. 2011. CS1 одржавање: Вишеструка имена: списак аутора (веза)
10. ^ Gale JD, Grossman CJ, Whitehead, JW Oxford AW, Bunce KT, Humphrey PP (1994). „GR113808: a novel, selective antagonist with high affinity at the 5-HT4 receptor.”. British Journal of Pharmacology. 111 (1): 332—8. PMC 1910004 . PMID 8012715. doi:10.1111/j.1476-5381.1994.tb14064.x. CS1 одржавање: Вишеструка имена: списак аутора (веза)
11. ^ Xu R, Hong J, Morse CL, Pike VW (2010-10-14). „Synthesis, structure-affinity relationships, and radiolabeling of selective high-affinity 5-HT4 receptor ligands as prospective imaging probes for positron emission tomography”. J Med Chem. 53 (19): 7035—47. PMC 2951497 . PMID 20812727. doi:10.1021/jm100668r. 

• Cecilie Löe Licht, Changes in the 5-HT₄ receptor in animal models of depression and antidepressant treatment, PhD thesis, Faculty of Health Sciences, University of Copenhagen. Submitted 2008 October.
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• Claeysen, S; Faye P; Sebben M; et al. (1997). „Cloning and expression of human 5-HT4S receptors. Effect of receptor density on their coupling to adenylyl cyclase.” (PDF). NeuroReport. 8 (15): 3189—96. PMID 9351641. S2CID 20624532. doi:10.1097/00001756-199710200-00002. 
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• Claeysen, S; Sebben M; Becamel C; et al. (1999). „Novel brain-specific 5-HT4 receptor splice variants show marked constitutive activity: role of the C-terminal intracellular domain.”. Mol. Pharmacol. 55 (5): 910—20. PMID 10220570. 
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• Medhurst, AD; Lezoualc'h F; Fischmeister R; et al. (2001). „Quantitative mRNA analysis of five C-terminal splice variants of the human 5-HT4 receptor in the central nervous system by TaqMan real time RT-PCR.”. Brain Res. Mol. Brain Res. 90 (2): 125—34. PMID 11406291. doi:10.1016/S0169-328X(01)00095-X. 
• Hiroi, T; Hayashi-Kobayashi N; Nagumo S; et al. (2002). „Identification and characterization of the human serotonin-4 receptor gene promoter.”. Biochem. Biophys. Res. Commun. 289 (2): 337—44. PMID 11716477. doi:10.1006/bbrc.2001.5979. 
• Vilaró MT, Doménech T, Palacios JM, Mengod G (2002). „Cloning and characterization of a novel human 5-HT4 receptor variant that lacks the alternatively spliced carboxy terminal exon. RT-PCR distribution in human brain and periphery of multiple 5-HT4 receptor variants.”. Neuropharmacology. 42 (1): 60—73. PMID 11750916. S2CID 23722311. doi:10.1016/S0028-3908(01)00154-X. 
• López-Rodríguez ML; Murcia M; Benhamú B; et al. (2002). „Computational model of the complex between GR113808 and the 5-HT4 receptor guided by site-directed mutagenesis and the crystal structure of rhodopsin.”. J. Comput. Aided Mol. Des. 15 (11): 1025—33. PMID 11989623. S2CID 23478175. doi:10.1023/A:1014895611874. 
• Ohtsuki, T; Ishiguro H; Detera-Wadleigh SD; et al. (2003). „Association between serotonin 4 receptor gene polymorphisms and bipolar disorder in Japanese case-control samples and the NIMH Genetics Initiative Bipolar Pedigrees.”. Mol. Psychiatry. 7 (9): 954—61. PMID 12399948. S2CID 21064320. doi:10.1038/sj.mp.4001133. 
• Norum JH, Hart K, Levy FO (2003). „Ras-dependent ERK activation by the human G(s)-coupled serotonin receptors 5-HT4(b) and 5-HT7(a).”. J. Biol. Chem. 278 (5): 3098—104. PMID 12446729. doi:10.1074/jbc.M206237200 . 
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• Cartier, D; Lihrmann I; Parmentier F; et al. (2003). „Overexpression of serotonin4 receptors in cisapride-responsive adrenocorticotropin-independent bilateral macronodular adrenal hyperplasia causing Cushing's syndrome.”. J. Clin. Endocrinol. Metab. 88 (1): 248—54. PMID 12519861. S2CID 40285098. doi:10.1210/jc.2002-021107. 
• Manzke, T; Guenther U; Ponimaskin, EG; et al. (2003). „5-HT4(a) receptors avert opioid-induced breathing depression without loss of analgesia.”. Science. 301 (5630): 226—9. Bibcode:2003Sci...301..226M. PMID 12855812. S2CID 13641423. doi:10.1126/science.1084674.